Mechanism of Action

Trestolone Acetate binds to androgen receptors in muscle and other tissues, activating pathways that promote muscle protein synthesis. This results in increased muscle mass, strength, and overall physical performance. It may also reduce muscle breakdown and support faster recovery.

Indications

Trestolone Acetate is indicated for testosterone replacement therapy in individuals with low testosterone levels. It may also be used in certain controlled athletic or bodybuilding contexts to support muscle growth and physical performance, although such use carries legal and ethical considerations.

Contraindications

Use of Trestolone Acetate is contraindicated in individuals with:

• Known hypersensitivity to Trestolone or any component of the formulation

• Prostate cancer or male breast cancer

• Significant cardiac, liver, or kidney disorders

Precautions

Caution is advised for patients with pre-existing liver, cardiovascular, or endocrine conditions. Regular monitoring of hormone levels, liver function, and other relevant clinical parameters is essential during treatment.

Drug Interactions

Trestolone Acetate may interact with medications affecting liver enzyme activity, altering its clearance. Concurrent use of other anabolic or androgenic agents may increase the risk of adverse effects. A full review of current medications is recommended before initiating therapy.

Dosage

Dosages vary depending on the indication and individual response:

• Performance enhancement: 50–200 mg per week, intramuscularly

• Therapeutic use: Determined by a healthcare provider based on clinical needs

Injection Site Care & Technique

• Warm the vial to body temperature before use

• Use a sterile 25G–27G needle and syringe

• Inject slowly to minimize tissue irritation

• Gently massage the site after injection

• Rotate injection sites to prevent tissue damage

• Avoid inflamed or previously used areas

• Keep the vial upright and avoid excessive agitation

Storage

Store at room temperature in a dry, dark place. Do not refrigerate. Keep out of reach of children.

Regulatory Compliance and Safety

• Manufactured according to Good Manufacturing Practices (GMP)

• Prescription-only medication, to be used under licensed medical supervision

• Report any adverse reactions to a healthcare provider

• Seek immediate medical attention in the event of an overdose